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Discovery of 5-Nitro-6-thiocyanatopyrimidines as Inhibitors of Cryptococcus  neoformans and Cryptococcus gattii | ACS Medicinal Chemistry Letters
Discovery of 5-Nitro-6-thiocyanatopyrimidines as Inhibitors of Cryptococcus neoformans and Cryptococcus gattii | ACS Medicinal Chemistry Letters

ACS Medicinal Chemistry Letters | Vol 11, No 11
ACS Medicinal Chemistry Letters | Vol 11, No 11

LogD Contributions of Substituents Commonly Used in Medicinal Chemistry |  ACS Medicinal Chemistry Letters
LogD Contributions of Substituents Commonly Used in Medicinal Chemistry | ACS Medicinal Chemistry Letters

Metabolically Stable tert-Butyl Replacement | ACS Medicinal Chemistry  Letters
Metabolically Stable tert-Butyl Replacement | ACS Medicinal Chemistry Letters

Supramolecular Self-Assembly To Control Structural and Biological  Properties of Multicomponent Hydrogels | Chemistry of Materials
Supramolecular Self-Assembly To Control Structural and Biological Properties of Multicomponent Hydrogels | Chemistry of Materials

Discovery of Novel Cyanamide-Based Inhibitors of Cathepsin C | ACS  Medicinal Chemistry Letters
Discovery of Novel Cyanamide-Based Inhibitors of Cathepsin C | ACS Medicinal Chemistry Letters

Myeloid Differentiation Primary Response Protein 88 (MyD88): The Central  Hub of TLR/IL-1R Signaling | Journal of Medicinal Chemistry
Myeloid Differentiation Primary Response Protein 88 (MyD88): The Central Hub of TLR/IL-1R Signaling | Journal of Medicinal Chemistry

Publications - The Frantz Lab
Publications - The Frantz Lab

Class 1 PI3K Clinical Candidates and Recent Inhibitor Design Strategies: A  Medicinal Chemistry Perspective | Journal of Medicinal Chemistry
Class 1 PI3K Clinical Candidates and Recent Inhibitor Design Strategies: A Medicinal Chemistry Perspective | Journal of Medicinal Chemistry

Discovery of a Selective Phosphoinositide-3-Kinase (PI3K)-γ Inhibitor  (IPI-549) as an Immuno-Oncology Clinical Candidate | ACS Medicinal  Chemistry Letters
Discovery of a Selective Phosphoinositide-3-Kinase (PI3K)-γ Inhibitor (IPI-549) as an Immuno-Oncology Clinical Candidate | ACS Medicinal Chemistry Letters

Discovery of APD371: Identification of a Highly Potent and Selective CB2  Agonist for the Treatment of Chronic Pain | ACS Medicinal Chemistry Letters
Discovery of APD371: Identification of a Highly Potent and Selective CB2 Agonist for the Treatment of Chronic Pain | ACS Medicinal Chemistry Letters

Robust and Tunable Hybrid Hydrogels from Photo-Cross-Linked Soy Protein  Isolate and Regenerated Silk Fibroin | ACS Sustainable Chemistry &  Engineering
Robust and Tunable Hybrid Hydrogels from Photo-Cross-Linked Soy Protein Isolate and Regenerated Silk Fibroin | ACS Sustainable Chemistry & Engineering

Structure–Activity Relationships of (+)-Naltrexone-Inspired Toll-like  Receptor 4 (TLR4) Antagonists | Journal of Medicinal Chemistry
Structure–Activity Relationships of (+)-Naltrexone-Inspired Toll-like Receptor 4 (TLR4) Antagonists | Journal of Medicinal Chemistry

a-Factor Analogues Containing Alkyne- and Azide-Functionalized Isoprenoids  Are Efficiently Enzymatically Processed and Retain Wild-Type Bioactivity |  Bioconjugate Chemistry
a-Factor Analogues Containing Alkyne- and Azide-Functionalized Isoprenoids Are Efficiently Enzymatically Processed and Retain Wild-Type Bioactivity | Bioconjugate Chemistry

Metabolically Stable tert-Butyl Replacement | ACS Medicinal Chemistry  Letters
Metabolically Stable tert-Butyl Replacement | ACS Medicinal Chemistry Letters

Sortase A Inhibitors: Recent Advances and Future Perspectives | Journal of  Medicinal Chemistry
Sortase A Inhibitors: Recent Advances and Future Perspectives | Journal of Medicinal Chemistry

Applications of Deuterium in Medicinal Chemistry | Journal of Medicinal  Chemistry
Applications of Deuterium in Medicinal Chemistry | Journal of Medicinal Chemistry

Metabolically Stable tert-Butyl Replacement | ACS Medicinal Chemistry  Letters
Metabolically Stable tert-Butyl Replacement | ACS Medicinal Chemistry Letters

Minor Structural Change to Tertiary Sulfonamide RORc Ligands Led to  Opposite Mechanisms of Action | ACS Medicinal Chemistry Letters
Minor Structural Change to Tertiary Sulfonamide RORc Ligands Led to Opposite Mechanisms of Action | ACS Medicinal Chemistry Letters

Discovery of a Novel Series of 7-Azaindole Scaffold Derivatives as PI3K  Inhibitors with Potent Activity | ACS Medicinal Chemistry Letters
Discovery of a Novel Series of 7-Azaindole Scaffold Derivatives as PI3K Inhibitors with Potent Activity | ACS Medicinal Chemistry Letters

Discovery of Highly Isoform Selective Thiazolopiperidine Inhibitors of  Phosphoinositide 3-Kinase γ | Journal of Medicinal Chemistry
Discovery of Highly Isoform Selective Thiazolopiperidine Inhibitors of Phosphoinositide 3-Kinase γ | Journal of Medicinal Chemistry

Publications - The Frantz Lab
Publications - The Frantz Lab

Dehydrozingerone Inspired Styryl Hydrazine Thiazole Hybrids as Promising  Class of Antimycobacterial Agents | ACS Medicinal Chemistry Letters
Dehydrozingerone Inspired Styryl Hydrazine Thiazole Hybrids as Promising Class of Antimycobacterial Agents | ACS Medicinal Chemistry Letters

Journal of Natural Products Special Issue Honors Drs. Rachel Mata and  Barbara N. Timmermann - ACS Axial
Journal of Natural Products Special Issue Honors Drs. Rachel Mata and Barbara N. Timmermann - ACS Axial